I-Pitavastatin Calcium

Incazelo emfushane:

Igama le-API Inkomba Ukucaciswa I-US DMF I-EU DMF CEP
I-Pitavastatin Calcium I-Hypercholesterolemia Endlini      


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

IMINININGWANE YOMKHIQIZO

匹伐他汀钙 I-Pitavastatin 147526-32-7 Endlini
PI-5 3800-06-4 Endlini
PI-6 145516-11-4 Endlini
PI-7 121660-11-5 Endlini

 

Incazelo

I-Pitavastatin Calcium (NK-104 hemicalcium) iyi-hydroxymethylglutaryl-CoA (HMG-CoA) reductase inhibitor enamandla.I-Pitavastatin Calcium (NK-104 hemicalcium) ivimbela ukwakheka kwe-cholesterol ku-acetic acid nge-IC50 ka-5.8 nM kumaseli e-HepG2.I-Pitavastatin Calcium iyi-hepatocyte low-density lipoprotein-cholesterol (LDL-C) receptor inducer esebenzayo.Umsebenzi wokulwa nomdlavuza.

 

Ingemuva

I-Pitavastatin Calcium iyi-inhibitor encintisanayo ye-enzyme HMGCR (HMG-CoA reductase) iphumela ekuncipheni kwe-LDL cholesterol synthesis.Olunye ucwaningo lubonisa ukuthi i-pitavastatin ingacindezela ukukhiqizwa komoyampilo kumaseli e-endothelial ngokuvimbela i-NADPH oxidase.Ngaphezu kwalokho, i-pitavastatin yehlisa ukuvezwa kwe-eNOS mRNA ngenkathi ikhulisa impendulo encike ku-NO egqugquzelwa i-acetylcholine ne-calcium ionophore, A23187.Ngaphezu kwalokho, i-pitavastatin ivimbela ukulawulwa kwe-conductance calcium-activated potassium channels ngokwehlisa amazinga e-cholesterol kumaseli.

 

Isitoreji

4°C, vikela ekukhanyeni

*Ku-solvent : -80°C, izinyanga ezingu-6;-20°C, inyanga engu-1 (vikela ekukhanyeni)

 

Isakhiwo samakhemikhali

Pitavastatin Calcium

Idatha Yebhayoloji Ehlobene

Pitavastatin Calcium2

ISItifiketi

2018 GMP-2
原料药GMP证书201811(captopril ,thalidomide etc)
GMP-of-PMDA-in-Chanyoo-平成28年08月03日 Nantong-Chanyoo-Pharmatech-Co
FDA-EIR-Letter-201901

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